a 92 — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T11373	GCN2-IN-1	A-92	Others
	GCN2-IN-1 (A-92) is an effective GCN2 inhibitor and can be used in research on the treatment of cancer as a chemotherapeutic agent.		Others
TPL0366	4-Biphenylcarboxylic acid
	4-Biphenylcarboxylic acid is a useful organic compound for research related to life sciences. The catalog number is TPL0366 and the CAS number is 92-92-2.
T28182	NNC 92-1687	NNC92-1687,NNC-92-1687	Glucagon Receptor
	NNC 92-1687 is a selective glucagon receptor antagonist that can be used to study type 2 diabetes.		Glucagon Receptor
T8922	SRS11-92	AA9	Ferroptosis
	SRS11-92 (AA9) is a ferroptosis inhibitor and a derivative of ferrostatin-1		Ferroptosis
T11805	L-NIL		Others
	L-NIL is a potent and selective inhibitor of inducible NO synthase with IC50s of 92 and 3.3 μM for rat brain constitutive NO synthase and mouse inducible NO synthase, respectively.		Others
T9223	RO-0335		Reverse Transcriptase
	RO-0335 is a potent diphenylether nonnucleoside reverse transcriptase inhibitor. RO-0335 inhibits Wt HIV-1 (IC50 = 1.1 nM) and retained activity (IC50< 100 nM) against 92% of a large number of NNRTI-resistant clinical is...		Reverse Transcriptase
T7214	TEPP-46	ML265	PKM
	TEPP-46 (ML265) is a potent PKM2 activator (AC50 : 92 nM) showing little or no effect on PKM1, PKL and PKR,induces tetramerization and reduces tumor formation and size in a mouse xenograft model. .		PKM
T21766	ML352
	ML352, a noncompetitive inhibitor of the presynaptic choline transporter (CHT), exhibits K i values of 92 nM in HEK293 cells with human CHT expression and 166 nM in mouse forebrain synaptosomes [1].
T9417L	Gamma-preprotachykinin amide (72-92) acetate	gamma-preprotachykinin amide (72-92) acetate (114882-65-4 Free base)	Others
	gamma-preprotachykinin amide (72-92) acetate is a 21 amino acid peptide belonging to the tachykinin (TK) family and including neurokinin A (NKA) in its C-terminal sequence. gamma-preprotachykinin amide (72-92) acetate po...		Others
T4530	KN-92 phosphate	KN92-H3PO4	CaMK
	KN-92 phosphate (KN92-H3PO4) is an inactive derivative of KN-93. KN-93 is a selective inhibitor of Ca2+/calmodulin-dependent kinase II (CaMKII), competitively blocking CaM binding to the kinase (Ki = 370 nM).		CaMK
T8543	KN-92 hydrochloride		CaMK
	KN-92 hydrochloride is an inactive derivative of KN-93. KN-93 is a selective Ca2+/calmodulin-dependent kinase II (CaMKII) inhibitor, competitively blocking CaM binding to the kinase with Ki of 370 nM.		CaMK
T8884	HSMG-1 inhibitor 11j		PI3K , mTOR
	hSMG-1 inhibitor 11j is a pyrimidine derivative. hSMG-1 inhibitor 11j is a potent and selective inhibitor of hSMG-1, IC50 = 0.11 nM. hSMG-1 inhibitor 11j exhibits >455-fold selectivity for hSMG-1 over mTOR (IC50=50 nM), ...		PI3K , mTOR
T8944	TTA-A2		Calcium Channel
	TTA-A2 is a selective T-type calcium channel antagonist as a potent anticonvulsant that the Cav3.1 isoform plays a prominent role in mediating. TTA-A2 is equally potent against the Cav3.1 (a1G) and Cav3.2 (a1H) channels ...		Calcium Channel
T4108	3-TYP	3-(1H-1,2,3-triazol-4-yl) pyridine	Sirtuin
	3-TYP (3-(1H-1,2,3-triazol-4-yl) pyridine) is a selective SIRT3 inhibitor.		Sirtuin
T6032	Birabresib	OTX-015,OTX015 （MK 8628/Birabresib）,MK-8628	Epigenetic Reader Domain
	Birabresib (MK-8628) is a synthetic, small molecule inhibitor of the BET (Bromodomain and Extra-Terminal) family of bromodomain-containing proteins 2, 3 and 4 with potential antineoplastic activity.		Epigenetic Reader Domain
T8756	KRAS inhibitor-9	DUN09716	Apoptosis , Ras
	KRAS inhibitor-9 (DUN09716) is a potent KRAS inhibitor with Kd of 92 μM that blocks the formation of GTP-KRAS and downstream activation of KRAS. KRAS inhibitor-9 causes G2/M cell cycle arrest and induces apoptosis. KRAS ...		Apoptosis , Ras
T36944	Ara-G		Nucleoside Antimetabolite/Analog
	Ara-G is an analog of the nucleoside guanosine and an active metabolite of nelarabine .1,2 Ara-G accumulates in T lymphoblasts and malignant T-lymphoid cells, where it is phosphorylated to produce ara-GTP and incorporate...		Nucleoside Antimetabolite/Analog
TP1488	Proadrenomedullin (45-92), human
	Proadrenomedullin (45-92), human, a mid-regional fragment of proadrenomedullin (MR-proADM), comprises amino acids 45–92 of pre-proADM.
T72350	Antibacterial agent 92
	Antibacterial agent 92, a triple-site aminoacyl-tRNA synthetase (aaRS) inhibitor, demonstrates a potent antibacterial effect by inhibiting Salmonella enterica threonyl-tRNA synthetase (SeThrRS) with an IC50 of 0.58 μM.
T70693	MRT-92 HCl salt
	MRT-92 is a potent and selective Smoothened (Smo) receptor inhibitor. MRT-92 displays subnanomolar antagonist activity against Smo in various Hh cell-based assays. MRT-92 inhibits rodent cerebellar granule cell prolifera...